SCHEMBL5633633

SCHEMBL5633633

O=C(O)c1cn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c(-c2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.53
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
TACR1 P25103 10/20 0.43
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ICMT O60725 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5632658 0.88 KDM4E (0.44) BRD4ALDH1A1TACR1KMT2AKDM4E
SCHEMBL4419725 0.83 BRD4 (0.67) BRD4ALDH1A1GAASMN1; SMN2
SCHEMBL4637805 0.78 GAA (0.52) ALDH1A1GAATACR1KDM4EHTT
SCHEMBL4638473 0.73 ALDH1A1 (0.65) ALDH1A1GAASMN1; SMN2POLB
Trifluoroacetic Acid SCHEMBL4737901 0.72 BRD4 (0.51) BRD4GAAPOLB
SCHEMBL4638859 0.71 SMN1; SMN2 (0.43) ALDH1A1GAATACR1KMT2AKDM4E
SCHEMBL4639437 0.71 TACR1 (0.43) ALDH1A1GAATACR1
SCHEMBL20603196 0.70 L3MBTL1 (0.57) ALDH1A1GAAKMT2AKDM4EHTT
SCHEMBL30379055 0.70 L3MBTL1 (0.57) ALDH1A1GAAKMT2AKDM4EHTT
SCHEMBL4706776 0.70 ALDH1A1 (0.54) ALDH1A1GAASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179804-B2 Tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 2007-02-20 US disclosed
US-20050239776-A1 Tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 2005-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050239776-A1 Tachykinin receptor antagonists TACR2, TACR1, PROKR1 BRD4 4297/4885ALDH1A1 1988/4885GAA 1920/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.