SCHEMBL5635294

SCHEMBL5635294

CCOC(=O)Cc1nc(Cc2ccccc2)no1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
L3MBTL1 Q9Y468 3/20 0.48
MAPT P10636 3/20 0.48
RXFP1 Q9HBX9 2/20 0.48
PRNP P04156 1/20 0.48
LMNA P02545 5/20 0.47
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
GLA P06280 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.44
CHUK O15111 1/20 0.43
TXNRD1 Q16881 1/20 0.43
NOX4 Q9NPH5 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11553918 0.82 MAPK1 (0.54) SMN1; SMN2L3MBTL1MAPTLMNAMAPK1
SCHEMBL553588 0.78 KLKB1 (0.49) SMN1; SMN2L3MBTL1MAPTRXFP1PRNP
SCHEMBL5634485 0.77 LMNA (0.44) SMN1; SMN2L3MBTL1MAPTLMNAALDH1A1
SCHEMBL28987843 0.77 SMN1; SMN2 (0.67) SMN1; SMN2L3MBTL1MAPTTSHRALDH1A1
SCHEMBL92379 0.77 MAPK1 (0.57) SMN1; SMN2L3MBTL1MAPTLMNAMAPK1
SCHEMBL562969 0.76 LMNA (0.46) SMN1; SMN2L3MBTL1MAPTRXFP1PRNP
SCHEMBL8132473 0.76 SMN1; SMN2 (0.52) SMN1; SMN2L3MBTL1MAPTRXFP1PRNP
SCHEMBL11550439 0.76 ALDH1A1 (0.55) SMN1; SMN2L3MBTL1MAPTLMNAMAPK1
SCHEMBL20020153 0.75 SMN1; SMN2 (0.38) SMN1; SMN2MAPK1TSHR
SCHEMBL10264767 0.74 MAPK1 (0.55) SMN1; SMN2L3MBTL1MAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
CN-1150192-C Piperidines as CCR5 modulators 2004-05-19 CN disclosed
CN-1331691-A Piperidines as CCR5 modulators PFIZER LTD (US) 2002-01-16 CN disclosed