SCHEMBL5635829

SCHEMBL5635829

COc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCCO3)c(C=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.38
THRB P10828 2/20 0.38
MAPT P10636 2/20 0.38
USP30 Q70CQ3 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
ALDH1A1 P00352 2/20 0.36
STS P08842 2/20 0.36
HTT P42858 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GPR119 Q8TDV5 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635973 0.92 STS (0.41) TP53THRBMAPTUSP30HTR2A
SCHEMBL5636701 0.91 USP30 (0.39) TP53THRBMAPTUSP30HTR2A
SCHEMBL5636737 0.90 USP30 (0.38) TP53THRBMAPTUSP30HTR2A
SCHEMBL5668341 0.90 MAPT (0.40) TP53THRBMAPTUSP30HTR2A
SCHEMBL5636475 0.90 USP30 (0.44) MAPTUSP30GPR119
SCHEMBL5636970 0.89 THRB (0.38) TP53THRBMAPTUSP30HTR2A
SCHEMBL5637216 0.89 HTR2A (0.49) TP53THRBMAPTUSP30HTR2A
SCHEMBL5848505 0.87 HTR2A (0.48) TP53HTR2AHTR2CHTR2BALDH1A1
SCHEMBL5848188 0.87 HTR2A (0.50) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5637246 0.86 USP30 (0.41) TP53THRBMAPTUSP30ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed