SCHEMBL5637246

SCHEMBL5637246

COc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCO3)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.41
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
PIK3CA P42336 3/20 0.39
ALDH1A1 P00352 3/20 0.38
STS P08842 1/20 0.38
PRKDC P78527 2/20 0.38
MTOR P42345 1/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GPR119 Q8TDV5 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636701 0.95 USP30 (0.39) USP30MAPTTP53THRBPIK3CA
SCHEMBL5637496 0.90 HTR2A (0.47) USP30MAPTTP53THRBPIK3CA
SCHEMBL5635973 0.88 STS (0.41) USP30MAPTTP53THRBALDH1A1
SCHEMBL5668341 0.87 MAPT (0.40) USP30MAPTTP53THRBALDH1A1
SCHEMBL5636737 0.87 USP30 (0.38) USP30MAPTTP53THRBALDH1A1
SCHEMBL5636970 0.86 THRB (0.38) USP30MAPTTP53THRBALDH1A1
SCHEMBL5635829 0.86 TP53 (0.38) USP30MAPTTP53THRBALDH1A1
SCHEMBL5847114 0.86 HTR2A (0.45) PIK3CAALDH1A1STSPRKDCMTOR
SCHEMBL5637216 0.85 HTR2A (0.49) USP30MAPTTP53THRBPIK3CA
SCHEMBL5637468 0.85 ALDH1A1 (0.39) PIK3CAALDH1A1STSPRKDCMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed