SCHEMBL5635897

SCHEMBL5635897

O=C(O)c1ccc2[nH]c(-c3ccc(-c4ccccn4)cc3)nc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 5/20 0.66
KDM4E B2RXH2 3/20 0.59
HPGD P15428 3/20 0.59
ALDH1A1 P00352 2/20 0.59
KMT2A Q03164 2/20 0.59
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
TGFBR1 P36897 2/20 0.56
SCD O00767 1/20 0.54
AURKA O14965 1/20 0.52
NR4A2 P43354 1/20 0.52
DHODH Q02127 2/20 0.52
PARP1 P09874 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
ACVR1B P36896 1/20 0.52
LMNA P02545 2/20 0.51
PKM P14618 2/20 0.51
MAPT P10636 1/20 0.51
FHIT P49789 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL179109 0.90 METAP2 (0.60) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL3921720 0.89 CHEK2 (0.83) CHEK2KDM4EHPGDALDH1A1TGFBR1
SCHEMBL3560621 0.86 KDM4E (0.66) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL8611783 0.86 KDM4E (0.69) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL28930292 0.85 KDM4E (0.68) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL7602620 0.84 KDM4E (0.70) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL1664016 0.83 MMP2 (0.66) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL11034496 0.81 METAP1 (0.58) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL20982594 0.80 NR4A2 (0.77) CHEK2KDM4EHPGDALDH1A1KMT2A
SCHEMBL6220033 0.80 PKN1 (0.60) CHEK2KDM4EHPGDALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271261-B2 Substituted benzimidazoles and imidazo-[4,5]-pyridines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2007-09-18 US claimed
US-7271261-B2 Substituted benzimidazoles and imidazo-[4,5]-pyridines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2007-09-18 US disclosed