SCHEMBL5636068

SCHEMBL5636068

COc1ccc(Nc2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCCS3)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.39
DRD2 P14416 11/20 0.39
HTR2A P28223 11/20 0.39
ALDH1A1 P00352 1/20 0.39
JAK3 P52333 2/20 0.39
JAK2 O60674 1/20 0.39
PTK2 Q05397 1/20 0.39
USP30 Q70CQ3 1/20 0.38
STS P08842 1/20 0.37
EPHX2 P34913 1/20 0.37
LCK P06239 1/20 0.36
BTK Q06187 1/20 0.36
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
PRKDC P78527 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637851 0.92 PIK3CA (0.43) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL5638812 0.87 DRD2 (0.44) HTR2CDRD2HTR2AJAK2
SCHEMBL6756119 0.86 HTR2C (0.42) HTR2CDRD2HTR2AALDH1A1JAK3
SCHEMBL5638464 0.83 ALDH1A1 (0.39) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL5635052 0.81 ALDH1A1 (0.38) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL5637649 0.80 HTR2C (0.58) HTR2CDRD2HTR2A
SCHEMBL6754171 0.80 HTT (0.38) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL5636090 0.79 HTR2C (0.37) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL6756093 0.79 EPHX2 (0.38) HTR2CDRD2HTR2AALDH1A1STS
SCHEMBL5637120 0.79 DRD2 (0.44) HTR2CDRD2HTR2AALDH1A1USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed