SCHEMBL5636828

SCHEMBL5636828

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3cc(Cl)ccc3Cl)cc3c1N2CCCO3

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.40
CNR1 P21554 2/20 0.39
PAK1 Q13153 1/20 0.37
MAPT P10636 3/20 0.37
TP53 P04637 3/20 0.36
GPR119 Q8TDV5 1/20 0.36
CNR2 P34972 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
UTS2R Q9UKP6 2/20 0.35
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
LMNA P02545 1/20 0.35
STS P08842 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636262 0.94 CNR1 (0.41) USP30CNR1PAK1MAPTTP53
SCHEMBL5637027 0.91 USP30 (0.46) USP30CNR1MAPTTP53CNR2
SCHEMBL5636742 0.91 USP30 (0.41) USP30CNR1PAK1MAPTTP53
SCHEMBL5636142 0.89 USP30 (0.44) USP30CNR1MAPTTP53HPGD
SCHEMBL5636680 0.88 USP30 (0.43) USP30CNR1MAPTTP53MEN1
SCHEMBL5636737 0.87 USP30 (0.38) USP30MAPTTP53GPR119MEN1
SCHEMBL5635408 0.86 GPR119 (0.39) USP30MAPTGPR119STS
SCHEMBL5637776 0.86 USP30 (0.49) USP30CNR1MAPTTP53CNR2
SCHEMBL5846950 0.86 HTR2A (0.40) USP30CNR1PAK1MAPTTP53
SCHEMBL5847676 0.85 GPR119 (0.39) USP30CNR1PAK1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed