SCHEMBL5636200

SCHEMBL5636200

COc1ccc(-c2cc3c4c(c2)C2CCN(C(=O)OC(C)(C)C)CCC2N4CCCS3)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.45
ALDH1A1 P00352 3/20 0.39
STS P08842 2/20 0.39
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GPR119 Q8TDV5 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TP53 P04637 1/20 0.38
HTR2A P28223 2/20 0.38
HTR2B P41595 1/20 0.38
EPHX2 P34913 1/20 0.37
DYRK1A Q13627 1/20 0.35
MAPT P10636 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635065 0.91 ALDH1A1 (0.40) HTR2CALDH1A1STSHTTMEN1
SCHEMBL5637526 0.91 HTR2C (0.55) HTR2CALDH1A1STSMEN1KMT2A
SCHEMBL5638128 0.91 HTR2C (0.55) HTR2CALDH1A1STSMEN1KMT2A
SCHEMBL5636957 0.87 HTR2C (0.43) HTR2CHTR2ADRD2
SCHEMBL5636395 0.86 HTR2C (0.43) HTR2CALDH1A1MEN1KMT2AGPR119
SCHEMBL5634987 0.86 HTR2C (0.54) HTR2CALDH1A1MEN1KMT2AHPGD
SCHEMBL5636180 0.86 HTR2C (0.54) HTR2CALDH1A1MEN1KMT2AHPGD
SCHEMBL6754171 0.85 HTT (0.38) HTR2CALDH1A1STSHTTMEN1
SCHEMBL6756119 0.85 HTR2C (0.42) HTR2CALDH1A1STSHTTMEN1
SCHEMBL5636090 0.85 HTR2C (0.37) HTR2CALDH1A1STSHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed