SCHEMBL5636571

SCHEMBL5636571

COC(=O)/C=C\c1cc(OC)ccc1-c1cc2c3c(c1)[C@@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1N3CCCS2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
STS P08842 2/20 0.35
HTR2C P28335 7/20 0.34
HTR2A P28223 5/20 0.34
HTR2B P41595 1/20 0.34
DRD2 P14416 4/20 0.34
EPHX2 P34913 1/20 0.34
HTT P42858 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BACE1 P56817 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
SRC P12931 2/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6756112 1.00 ALDH1A1 (0.35) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5637381 0.92 HTR2C (0.35) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5636382 0.91 HTR2C (0.37) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636090 0.91 HTR2C (0.37) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5636083 0.91 HTR2C (0.37) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636162 0.90 HTR2C (0.36) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5635167 0.90 HTR2C (0.36) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5635106 0.90 HTR2C (0.36) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL5635052 0.87 ALDH1A1 (0.38) ALDH1A1STSHTR2CHTR2AHTR2B
SCHEMBL6754171 0.86 HTT (0.38) ALDH1A1STSHTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed