SCHEMBL5636952

SCHEMBL5636952

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(C3CCCC3)cc3c1N2CCCS3

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.40
HTR2C P28335 18/20 0.38
DRD2 P14416 17/20 0.38
HTR2A P28223 17/20 0.38
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635083 0.99 PDE4B (0.40) PDE4BHTR2CDRD2HTR2AKDM4E
SCHEMBL5639095 0.87 GPR119 (0.39) HTR2CDRD2HTR2A
SCHEMBL5637490 0.87 HTR2C (0.42) HTR2CDRD2HTR2A
SCHEMBL5637898 0.87 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5638532 0.87 HTR2C (0.39) PDE4BHTR2CDRD2HTR2A
SCHEMBL5636432 0.87 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5637177 0.87 HTR2C (0.42) HTR2CDRD2HTR2A
SCHEMBL5634923 0.87 HTR2C (0.43) HTR2CDRD2HTR2A
SCHEMBL5637123 0.86 HTR2C (0.37) PDE4BHTR2CDRD2HTR2A
SCHEMBL5638464 0.86 ALDH1A1 (0.39) PDE4BHTR2CDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed