SCHEMBL5637067

SCHEMBL5637067

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(/C=C/c3ccccc3Cl)cc3c1N2CCCS3

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.39
HTR2A P28223 16/20 0.39
HTR2C P28335 16/20 0.39
STS P08842 2/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635914 0.90 DRD2 (0.42) DRD2HTR2AHTR2C
SCHEMBL5637022 0.88 DRD2 (0.44) DRD2HTR2AHTR2CSTS
SCHEMBL5638593 0.88 HTR2C (0.43) DRD2HTR2AHTR2C
SCHEMBL5637446 0.85 HTR2C (0.43) DRD2HTR2AHTR2C
SCHEMBL5636706 0.84 STS (0.37) DRD2HTR2AHTR2CSTS
SCHEMBL5637179 0.84 HTR2C (0.38) DRD2HTR2AHTR2C
SCHEMBL5636679 0.84 HTR2C (0.38) DRD2HTR2AHTR2C
SCHEMBL5638054 0.83 HTR2C (0.47) DRD2HTR2AHTR2CSTS
SCHEMBL5635470 0.83 HTR2C (0.47) DRD2HTR2AHTR2CSTS
SCHEMBL5636086 0.79 USP30 (0.45) DRD2HTR2AHTR2CSTS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed