SCHEMBL5636706

SCHEMBL5636706

COc1ccc(/C=C/c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCCS3)c(C)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
STS P08842 2/20 0.37
ALDH1A1 P00352 1/20 0.35
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
PRKDC P78527 1/20 0.35
DRD2 P14416 11/20 0.35
HTR2A P28223 11/20 0.35
HTR2C P28335 11/20 0.35
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
PDE4B Q07343 1/20 0.34
EPHX2 P34913 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635914 0.85 DRD2 (0.42) DRD2HTR2AHTR2C
SCHEMBL5637067 0.84 DRD2 (0.39) STSDRD2HTR2AHTR2C
SCHEMBL5638464 0.83 ALDH1A1 (0.39) STSALDH1A1DRD2HTR2AHTR2C
SCHEMBL5637851 0.83 PIK3CA (0.43) STSALDH1A1PIK3CAMTORPRKDC
SCHEMBL5636090 0.82 HTR2C (0.37) STSALDH1A1DRD2HTR2AHTR2C
SCHEMBL5637446 0.82 HTR2C (0.43) DRD2HTR2AHTR2C
SCHEMBL5637022 0.82 DRD2 (0.44) STSDRD2HTR2AHTR2C
SCHEMBL5637179 0.82 HTR2C (0.38) DRD2HTR2AHTR2CPDE4BKDM4E
SCHEMBL5636679 0.82 HTR2C (0.38) DRD2HTR2AHTR2CPDE4BKDM4E
SCHEMBL5637381 0.81 HTR2C (0.35) STSALDH1A1DRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed