SCHEMBL5637688

SCHEMBL5637688

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(Br)cc3c1N2CCO3

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 6/20 0.42
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
PIK3CA P42336 2/20 0.37
HTR2A P28223 6/20 0.37
HTR2C P28335 6/20 0.37
DRD2 P14416 4/20 0.37
RECQL P46063 1/20 0.36
GPR119 Q8TDV5 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
THRB P10828 1/20 0.36
HTR1A P08908 1/20 0.36
DRD4 P21917 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635355 0.94 USP30 (0.40) USP30IDO1TDO2PIK3CAHTR2A
SCHEMBL5637607 0.94 USP30 (0.40) USP30IDO1TDO2PIK3CAHTR2A
SCHEMBL5635404 0.93 USP30 (0.39) USP30HTR2AHTR2CRECQLGPR119
SCHEMBL6491628 0.84 USP30 (0.42) USP30IDO1TDO2PIK3CAHTR2A
SCHEMBL6491629 0.84 USP30 (0.42) USP30IDO1TDO2PIK3CAHTR2A
SCHEMBL6756087 0.84 HTR2A (0.41) HTR2AHTR2CDRD2HTR1ADRD4
SCHEMBL5421540 0.82 USP30 (0.41) USP30IDO1TDO2HTR2AHTR2C
SCHEMBL5848252 0.82 USP30 (0.41) USP30IDO1TDO2HTR2AHTR2C
SCHEMBL5635971 0.82 USP30 (0.47) USP30HTR2AHTR2CDRD2MAPT
SCHEMBL5637776 0.81 USP30 (0.49) USP30HTR2AHTR2CDRD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed