Noroxyhydrastinine

Noroxyhydrastinine

SCHEMBL564339

O=C1NCCc2cc3c(cc21)OCO3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 1.00
PARP10 Q53GL7 13/20 0.49
PARP11 Q9NR21 9/20 0.49
PARP1 P09874 6/20 0.49
F7 P08709 1/20 0.49
F3 P13726 1/20 0.49
PDPK1 O15530 1/20 0.46
ACHE P22303 1/20 0.44
CYP2D6 P10635 1/20 0.42
GRM5 P41594 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Noroxyhydrastinine SCHEMBL29745981 1.00 KDM4E (1.00) KDM4EPARP10PARP11PARP1F7
SCHEMBL30142226 0.81 KDM4E (0.69) KDM4EPARP1ACHECYP2D6GRM5
SCHEMBL12745699 0.78 KDM4E (0.63) KDM4EPARP10PARP11ACHECYP2D6
SCHEMBL9739665 0.75 KDM4E (0.60) KDM4EPARP10PARP11PARP1ACHE
SCHEMBL9739248 0.75 KDM4E (0.59) KDM4EPARP10PARP11PARP1F7
SCHEMBL6488098 0.74 KDM4E (0.59) KDM4EACHECYP2D6
SCHEMBL6488102 0.74 KDM4E (0.59) KDM4EACHECYP2D6
SCHEMBL6488092 0.74 KDM4E (0.59) KDM4EACHECYP2D6
SCHEMBL5568453 0.73 KDM4E (0.58) KDM4ECYP2D6
SCHEMBL6336267 0.73 KDM4E (0.58) KDM4EACHECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11753431-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2023-09-12 US disclosed
US-11753431-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2023-09-12 US disclosed
US-20210388017-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF INTOCELL, INC. (KP) 2021-12-16 US disclosed
WO-2019008441-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF INTOCELL, INC. (KR) 2019-01-10 WO disclosed
CN-102908341-A Vitexicarpin used as pharmaceutical active ingredient with anti-angiogenesis function UNIV TSINGHUA 2013-02-06 CN disclosed
CN-102030812-B Timosaponin A-III serving as medicinal active ingredient with angiogenesis resistance UNIV TSINGHUA 2012-07-04 CN disclosed
US-20120035855-A1 METHOD OF NETWORK-BASED IDENTIFICATION FOR DRUG ACTION AND/OR SYNERGY EFFECT OF MEDICINE COMBINATION TSINGHUA UNIVERSITY 2012-02-09 US disclosed
EP-2369493-A1 GENE NETWORK-BASED METHOD FOR CONFIRMING DRUG ACTION Tsinghua University (CN) 2011-09-28 EP disclosed
CN-102030812-A Timosaponin A-III serving as medicinal active ingredient with angiogenesis resistance UNIV TSINGHUA 2011-04-27 CN disclosed
CN-102028679-A Vitexin as active ingredient of medicine with anti-angiogenesis effect UNIV TSINGHUA 2011-04-27 CN disclosed
US-20110086872-A1 Berberine as a selective lung cancer agent and other compositions and methods TIN-WA MAUNG 2011-04-14 US disclosed
US-20070298132-A1 Berberine as a selective lung cancer agent PHARMCHEM INC. (US) 2007-12-27 US disclosed
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210388017-A1 COMPOUNDS COMPRISING CLEAVABLE LINKER AND USES THEREOF VIP, ANTXR2, TNFRSF9 KDM4E 3750/4885PARP10 3044/4885PARP11 3705/4885
US-11753431-B2 Compounds comprising cleavable linker and uses thereof VIP, ANTXR2, TNFRSF9 KDM4E 3750/4885PARP10 3044/4885PARP11 3705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.