SCHEMBL5645124

SCHEMBL5645124

CC(CC#N)(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.49
CYP2C19 P33261 2/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
CYP2C9 P11712 1/20 0.49
NPY2R P49146 1/20 0.49
TAAR1 Q96RJ0 1/20 0.41
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
MAPK1 P28482 1/20 0.39
CYP3A4 P08684 2/20 0.38
HIF1A Q16665 1/20 0.38
ATM Q13315 1/20 0.37
ALDH1A1 P00352 3/20 0.37
ALOX15 P16050 1/20 0.37
MAPT P10636 2/20 0.36
KCNN4 O15554 3/20 0.35
ESR1 P03372 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11724581 0.82 CYP2C19 (0.47) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL4673742 0.82 TAAR1 (0.52) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL955513 0.78 CYP2C19 (0.42) CYP2D6CYP2C19KMT2ACYP2C9TAAR1
SCHEMBL9398476 0.78 ESR1 (0.50) KMT2AMEN1CYP3A4ALDH1A1ESR1
SCHEMBL11421695 0.78 TAAR1 (0.43) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL30338404 0.78 MAPT (0.39) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL31310650 0.78 CYP2C19 (0.42) CYP2D6CYP2C19KMT2ACYP2C9TAAR1
SCHEMBL30338355 0.78 CYP2A6 (0.33) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL5180038 0.77 CYP2C19 (0.49) CYP2D6CYP2C19KMT2AMEN1CYP2C9
SCHEMBL27819578 0.77 ALDH1A1 (0.50) CYP2D6CYP2C19KMT2AMEN1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103242214-B A kind of indole derivatives and preparation method thereof SHAANXI BUCHANG HIGH-TECH PHARMACEUTICAL CO., LTD. (CN) 2016-04-06 CN claimed
CN-103641938-B A kind of initiator that can be used for vinyl monomer polyreaction BEIJING UNIVERSITY OF CHEMICAL TECHNOLOGY (CN) 2015-10-28 CN claimed
CN-104668552-B A kind of aluminium powder for 3D printing and preparation method thereof 成都新柯力化工科技有限公司 2016-09-07 CN disclosed
CN-103242214-B A kind of indole derivatives and preparation method thereof SHAANXI BUCHANG HIGH-TECH PHARMACEUTICAL CO., LTD. (CN) 2016-04-06 CN disclosed
CN-105348564-A Preparation method of inorganic powder specially used for low-density composite ivory boards CHENGDU NEW KELI CHEM SCI CO 2016-02-24 CN disclosed
CN-103772286-B A kind of method preparing imidafenacin JIANGXI QINGFENG PHARMACEUTICAL CO., LTD. (CN) 2016-01-13 CN disclosed
CN-103772286-B A kind of method preparing imidafenacin JIANGXI QINGFENG PHARMACEUTICAL CO., LTD. (CN) 2016-01-13 CN disclosed
CN-103641938-B A kind of initiator that can be used for vinyl monomer polyreaction BEIJING UNIVERSITY OF CHEMICAL TECHNOLOGY (CN) 2015-10-28 CN disclosed
CN-104668552-A Aluminum powder for 3D (three-dimensional) printing and preparation method of aluminum powder CHENGDU NEW KELI CHEM SCI CO 2015-06-03 CN disclosed
US-7169924-B2 Pyrimidinone derivatives and their use in the treatment of atherosclerosis SMITHKLINE BEECHAM PLC (GB) 2007-01-30 US disclosed
EP-0892787-A1 NOVEL $g(a)-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1999-01-27 EP disclosed
WO-1997038981-A1 NOVEL α-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1997-10-23 WO disclosed
US-5266718-A Antidiabetic agents ADIR ET COMPAGNIE (FR) 1993-11-30 US disclosed
EP-0518769-A1 Ethanolaminebenzoate derivative, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-12-16 EP disclosed