SCHEMBL565044

SCHEMBL565044

CC(C)(C)OC(=O)NC1(CN2CCc3cc(O)ccc32)COC(C)(C)OC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.42
PDK1 Q15118 2/20 0.37
PDK2 Q15119 2/20 0.37
PDK3 Q15120 2/20 0.37
PDK4 Q16654 2/20 0.37
GPR119 Q8TDV5 3/20 0.36
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ALOX5 P09917 2/20 0.33
EPHX2 P34913 2/20 0.33
PPIA P62937 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
KCNT1 Q5JUK3 1/20 0.31
NQO2 P16083 1/20 0.31
NR1H2 P55055 1/20 0.31
ESR1 P03372 3/20 0.31
DRD2 P14416 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL564864 0.86 NOTUM (0.34) ESR2PDK1PDK2PDK3PDK4
SCHEMBL2478769 0.70 CA1 (0.40) ESR2MAPK1NR1H2DRD2
SCHEMBL565811 0.69 S1PR1 (0.58) NPC1MAPTRAB9A
SCHEMBL565919 0.69 CHRM2 (0.38) MAPT
SCHEMBL566357 0.69 THRB (0.45) MAPT
SCHEMBL566353 0.69 ESR2 (0.41) ESR2ESR1DRD2
SCHEMBL79673 0.69 TDP1 (0.35) MAPK1
SCHEMBL29169997 0.69 HCRTR2 (0.34) MAPK1
SCHEMBL16589978 0.69 ESR2 (0.32) ESR2
SCHEMBL3899182 0.68 ESR2 (0.61) ESR2PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9181182-B2 S1P receptors modulators AKAAL PHARMA PTY LTD (AU) 2015-11-10 US disclosed
US-20120034270-A1 S1P Receptors Modulators AKAAL PHARMA PTY LTD (AU) 2012-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120034270-A1 S1P Receptors Modulators S1PR1, S1PR5, S1PR3 ESR2 958/4885PDK1 689/4885PDK2 1856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.