SCHEMBL5653534

SCHEMBL5653534

CCCn1c(=O)c2c(nc(Cc3ccc(S(C)(=O)=O)cc3)n2CCNCC(O)CC)n(CCc2ccc(N)cc2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.41
ADORA2B P29275 8/20 0.39
ADORA2A P29274 8/20 0.39
ADORA3 P0DMS8 3/20 0.38
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1332529 0.91 ADORA1 (0.42) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1332404 0.91 ADORA2B (0.44) ADORA1ADORA2BADORA2AADORA3TSHR
Hydrochloric Acid SCHEMBL1332577 0.91 ADORA2B (0.43) ADORA1ADORA2BADORA2AADORA3TSHR
SCHEMBL1332763 0.89 ADORA1 (0.41) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1333085 0.88 ADORA1 (0.41) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL4176171 0.88 ADORA1 (0.41) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1332443 0.87 ADORA1 (0.40) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1334668 0.87 ADORA1 (0.42) ADORA1ADORA2BADORA2AADORA3TSHR
SCHEMBL1333189 0.86 ADORA3 (0.40) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1334307 0.86 ADORA2B (0.47) ADORA1ADORA2BADORA2AADORA3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247639-B2 A1 adenosine receptor antagonists ENDACEA, INC. (US) 2007-07-24 US claimed