SCHEMBL5656674

SCHEMBL5656674

COC(=O)CSc1ncc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 15/20 0.74
CXCR1 P25024 9/20 0.74
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
ATM Q13315 1/20 0.50
P4HTM Q9NXG6 1/20 0.49
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5660669 0.88 CXCR2 (0.76) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5659975 0.86 CXCR2 (0.73) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL5846271 0.85 CXCR2 (1.00) CXCR2CXCR1MAPT
SCHEMBL5660105 0.82 CXCR1 (0.58) CXCR2CXCR1MAPT
SCHEMBL5660018 0.81 CXCR2 (0.79) CXCR2CXCR1
SCHEMBL14587553 0.80 P4HTM (0.57) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5658349 0.80 CXCR2 (0.73) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5657748 0.79 CXCR2 (0.65) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL5846226 0.76 CXCR2 (1.00) CXCR2CXCR1
SCHEMBL6850672 0.75 CXCR2 (0.84) CXCR2CXCR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US claimed
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed