SCHEMBL5658799

SCHEMBL5658799

O=C(O)CCNc1ncc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 7/20 0.60
CXCR1 P25024 5/20 0.60
P4HTM Q9NXG6 2/20 0.54
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
EGLN2 Q96KS0 1/20 0.49
MITF O75030 1/20 0.49
CCNA2 P20248 1/20 0.48
CDK2 P24941 1/20 0.48
PTPN1 P18031 1/20 0.48
PTPN6 P29350 1/20 0.48
PTPN11 Q06124 1/20 0.48
ALDH1A1 P00352 1/20 0.47
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
KCNE1 P15382 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5656205 0.82 CXCR2 (0.53) CXCR2CXCR1P4HTMHDAC3HDAC1
SCHEMBL5657748 0.78 CXCR2 (0.65) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL2703268 0.76 POLB (0.61) HDAC3HDAC1HDAC2HDAC6NPC1
SCHEMBL5656328 0.76 P4HTM (0.57) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL5659975 0.75 CXCR2 (0.73) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL16436048 0.74 PTPN1 (0.61) CXCR2CXCR1P4HTMHDAC3HDAC1
SCHEMBL16436052 0.74 KCNQ3 (0.65) CXCR2P4HTMNPC1RAB9AMITF
SCHEMBL5845348 0.73 CXCR2 (0.89) CXCR2CXCR1
SCHEMBL5846781 0.73 CXCR2 (1.00) CXCR2CXCR1
SCHEMBL3064046 0.72 P4HTM (0.67) CXCR2CXCR1P4HTMNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US claimed
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed