SCHEMBL5656205

SCHEMBL5656205

CC(C)(C)OC(=O)CCNc1ncc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 14/20 0.53
CXCR1 P25024 13/20 0.53
CTNNB1 P35222 1/20 0.47
TCF7L2 Q9NQB0 1/20 0.47
P4HTM Q9NXG6 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5658799 0.82 CXCR2 (0.60) CXCR2CXCR1P4HTMALDH1A1HDAC3
SCHEMBL5659634 0.81 CXCR1 (0.58) CXCR2CXCR1CTNNB1TCF7L2P4HTM
SCHEMBL5846063 0.76 CXCR1 (0.79) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL9891433 0.73 HDAC8 (0.42) CTNNB1TCF7L2ALDH1A1HDAC3HDAC1
SCHEMBL8352922 0.72 L3MBTL1 (0.54) HDAC6
SCHEMBL5658349 0.70 CXCR2 (0.73) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL7080560 0.70 NAMPT (0.64)
SCHEMBL28466017 0.70 MAPT (0.50) ALDH1A1
SCHEMBL5660669 0.69 CXCR2 (0.76) CXCR2CXCR1P4HTM
SCHEMBL5930648 0.69 POLB (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed