SCHEMBL5659995

SCHEMBL5659995

Nc1nc(SCC(=O)OCc2ccc(Cl)cc2)ncc1C(=O)Nc1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 5/20 0.52
CXCR2 P25025 5/20 0.52
MAPT P10636 4/20 0.47
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
AHR P35869 1/20 0.44
HSD17B10 Q99714 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
KLK7 P49862 1/20 0.42
TSHR P16473 2/20 0.42
MAPK10 P53779 1/20 0.42
MAPK1 P28482 1/20 0.41
NR3C1 P04150 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5657939 0.91 CXCR2 (0.53) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5657929 0.89 CXCR1 (0.51) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5657932 0.88 CXCR2 (0.54) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5659346 0.88 ALDH1A1 (0.54) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5658611 0.86 CXCR1 (0.46) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5658497 0.85 LMNA (0.56) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5657757 0.84 ALDH1A1 (0.58) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5660079 0.83 SMN1; SMN2 (0.51) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5660105 0.83 CXCR1 (0.58) CXCR1CXCR2MAPTALDH1A1KDM4E
SCHEMBL5659631 0.83 CXCR1 (0.62) CXCR1CXCR2MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US claimed
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed