SCHEMBL5664722

SCHEMBL5664722

CC(CNC(=O)[CH]c1ccccn1)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 3/20 0.38
POLB P06746 2/20 0.38
ESR1 P03372 1/20 0.38
CYP1A2 P05177 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5664584 0.79 KDM4E (0.40) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL4989140 0.79 HTT (0.40) ALDH1A1POLBCYP1A2MAPTTSHR
SCHEMBL5664580 0.76 HDAC3 (0.45) ALDH1A1KDM4ECYP1A2SMN1; SMN2LMNA
SCHEMBL14152063 0.76 KDM4E (0.41) ALDH1A1KDM4ECYP1A2SMN1; SMN2MAPT
SCHEMBL5666957 0.75 HDAC3 (0.43) ALDH1A1KDM4ECYP1A2SMN1; SMN2L3MBTL1
SCHEMBL5665489 0.75 HDAC3 (0.50) ALDH1A1KDM4ECYP1A2SMN1; SMN2L3MBTL1
SCHEMBL5664191 0.74 HDAC3 (0.55) ALDH1A1KDM4ECYP1A2SMN1; SMN2HPGD
SCHEMBL1516264 0.73 NPC1 (0.45) ALDH1A1KDM4ECYP1A2SMN1; SMN2LMNA
SCHEMBL5665952 0.73 HDAC6 (0.57) ALDH1A1CYP1A2SMN1; SMN2CYP2C19HDAC3
SCHEMBL1515297 0.73 L3MBTL1 (0.54) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716137-A1 SUBSTITUTED QUINOLINE COMPOUNDS Pfizer Products Incorporated (US) 2006-11-02 EP disclosed
WO-2005080373-A1 SUBSTITUTED QUINOLINE COMPOUNDS PFIZER PRODUCTS INC. (US) 2005-09-01 WO disclosed