SCHEMBL5673194

SCHEMBL5673194

O=C(O)Nc1c(F)cccc1CN(Cc1ccccc1)C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 18/20 0.51
SLC6A3 Q01959 11/20 0.51
SLC6A4 P31645 14/20 0.46
DCUN1D1 Q96GG9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744569 0.80 DCUN1D1 (0.52) SLC6A2SLC6A3SLC6A4DCUN1D1
SCHEMBL2877349 0.75 SLC6A2 (0.73) SLC6A2SLC6A3SLC6A4
Hydrochloric Acid SCHEMBL15012233 0.71 SLC6A2 (0.57) SLC6A2SLC6A3SLC6A4
Hydrochloric Acid SCHEMBL15012232 0.71 SLC6A2 (0.57) SLC6A2SLC6A3SLC6A4
SCHEMBL4585074 0.70 SLC6A2 (0.52) SLC6A2SLC6A3SLC6A4
SCHEMBL3811903 0.68 DCUN1D1 (0.58) SLC6A2SLC6A3SLC6A4DCUN1D1
Hydrochloric Acid SCHEMBL22797970 0.68 SLC6A2 (0.59) SLC6A2SLC6A3SLC6A4DCUN1D1
SCHEMBL4585570 0.68 SLC6A2 (0.47) SLC6A2SLC6A3SLC6A4
SCHEMBL20475214 0.68 RAB9A (0.51)
Fumaric Acid SCHEMBL5439692 0.67 SLC6A2 (1.00) SLC6A2SLC6A3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730137-A1 HETEROCYCLIC CGRP ANTAGONISTS FOR THE TREATMENT OF MIGRAINE Bristol-Myers Squibb Company (US) 2006-12-13 EP disclosed
WO-2005095383-A1 HETEROCYCLIC CGRP ANTAGONISTS FOR THE TREATMENT OF MIGRAINE BRISTOL-MYERS SQUIBB COMPANY (US) 2005-10-13 WO disclosed