SCHEMBL5683290

SCHEMBL5683290

COc1ccc(-c2ccc3[nH]c(N)nc3c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 3/20 0.48
KDM4E B2RXH2 3/20 0.48
PKM P14618 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
RAB9A P51151 2/20 0.48
DYRK1A Q13627 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
MAP4K4 O95819 1/20 0.46
TYMS P04818 2/20 0.45
FABP6 P51161 1/20 0.45
PRKAG1 P54619 1/20 0.45
PRKAA1 Q13131 1/20 0.45
PRKAB1 Q9Y478 1/20 0.45
MASP2 O00187 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2163036 0.87 TYMS (0.52) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL5679580 0.87 MAP4K4 (0.49) ALDH1A1NPC1PKMSMN1; SMN2RAB9A
Bromide SCHEMBL17747821 0.85 TYMS (0.51) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL4323448 0.83 NPC1 (0.49) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL5679426 0.82 FABP6 (0.53) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL419326 0.81 NPC1 (0.71) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL5680087 0.81 TYMS (0.44) ALDH1A1NPC1KDM4EPKMSMN1; SMN2
SCHEMBL3827667 0.80 ALDH1A1 (0.58) ALDH1A1NPC1KDM4ESMN1; SMN2RAB9A
SCHEMBL14395105 0.80 LOXL2 (0.57) FABP6MAPT
Hydrochloric Acid SCHEMBL7240756 0.79 CCR1 (0.47) ALDH1A1NPC1PKMSMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620413-A2 COMPOUNDS, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2006-02-01 EP disclosed
WO-2004098494-A2 COMPOUNDS, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2004-11-18 WO disclosed