SCHEMBL5684491

SCHEMBL5684491

CCCCc1ccc2c(c1)Cc1cc(-c3cc(F)c(C#N)c(F)c3)ccc1-2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 2/20 0.38
KCNH2 Q12809 1/20 0.38
RARB P10826 3/20 0.38
RARA P10276 1/20 0.38
RARG P13631 1/20 0.38
MPL P40238 7/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HRH3 Q9Y5N1 1/20 0.33
DRD2 P14416 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
GRM2 Q14416 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
FASN P49327 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5684072 0.96 TSHR (0.42) KCNJ1KCNH2RARBRARARARG
SCHEMBL5684164 0.95 TSHR (0.44) KCNJ1KCNH2RARBRARARARG
SCHEMBL5684293 0.95 TSHR (0.44) KCNJ1KCNH2RARBRARARARG
SCHEMBL5683617 0.93 KCNJ1 (0.39) KCNJ1KCNH2RARBRARARARG
SCHEMBL5683868 0.88 RARB (0.34) KCNJ1KCNH2RARBRARARARG
SCHEMBL5884539 0.88 KCNJ1 (0.48) KCNJ1KCNH2RARBRARARARG
SCHEMBL5686441 0.88 KCNJ1 (0.39) KCNJ1KCNH2TSHRTRPV4FASN
SCHEMBL5683559 0.85 MPL (0.38) KCNJ1KCNH2RARBRARARARG
SCHEMBL5684136 0.85 RARB (0.38) KCNJ1KCNH2RARBRARARARG
SCHEMBL5687512 0.85 KCNJ1 (0.48) KCNJ1KCNH2RARBRARARARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed