SCHEMBL5685113

SCHEMBL5685113

CCOC(=O)c1cc2cccc(CO)c2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.59
CCNB1 P14635 1/20 0.59
RAB9A P51151 4/20 0.57
KDM4E B2RXH2 3/20 0.57
ALDH1A1 P00352 3/20 0.57
HPGD P15428 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
NPC1 O15118 2/20 0.57
LMNA P02545 2/20 0.57
MAPT P10636 2/20 0.57
MEN1 O00255 1/20 0.57
GLA P06280 1/20 0.57
GAA P10253 1/20 0.57
KMT2A Q03164 1/20 0.57
ATM Q13315 1/20 0.57
HSD17B10 Q99714 1/20 0.51
ALOX15 P16050 1/20 0.49
HTT P42858 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045458 0.92 RAB9A (0.59) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL28784003 0.87 RAB9A (0.52) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL28944811 0.86 RAB9A (0.51) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL5110272 0.86 GLA (0.50) CDK1CCNB1ALDH1A1HPGDLMNA
SCHEMBL2455047 0.85 KDM4E (0.53) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL27782467 0.85 RAB9A (0.50) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL31501839 0.84 KDM4E (0.61) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL4040141 0.84 KDM4E (0.61) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL27804111 0.83 RAB9A (0.51) CDK1CCNB1RAB9AKDM4EALDH1A1
SCHEMBL29291197 0.83 RAB9A (0.51) CDK1CCNB1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631567-A2 HETEROCYCLIC N-ARYL CARBOXAMIDES AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-03-08 EP disclosed
WO-2005016918-A2 HETEROCYCLIC N-ARYL CARBOXAMIDES AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-02-24 WO disclosed