SCHEMBL5685205

SCHEMBL5685205

CN1CCN(c2nccc(Oc3cccc4cc(C(=O)O)n(C)c34)n2)CC1.COc1ccc(C(C)(C)C)cc1N

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.38
BRAF P15056 3/20 0.37
PTK2 Q05397 2/20 0.37
GSK3A P49840 1/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAP4K1 Q92918 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047440 0.86 MAP3K7 (0.39) MAPK14PTK2ALDH1A1NPSR1HSD17B10
SCHEMBL5685202 0.85 BRAF (0.47) MAPK14BRAFPTK2GSK3AALDH1A1
SCHEMBL5682611 0.85 MAPK14 (0.52) MAPK14BRAFGSK3A
SCHEMBL5119462 0.82 MAPK14 (0.39) MAPK14PTK2ALDH1A1SMN1; SMN2NPSR1
SCHEMBL5125191 0.79 ACHE (0.43) MAPK14ALDH1A1NPSR1HSD17B10
SCHEMBL5114170 0.78 ACHE (0.36) MAPK14ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL13688795 0.77 BRAF (0.37) MAPK14BRAFPTK2GSK3A
SCHEMBL14276192 0.77 MAPK14 (0.45) MAPK14PTK2GSK3A
SCHEMBL13688769 0.77 MAPK14 (0.40) MAPK14BRAFPTK2
SCHEMBL13688785 0.76 MAPK14 (0.39) MAPK14BRAFPTK2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631567-A2 HETEROCYCLIC N-ARYL CARBOXAMIDES AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-03-08 EP claimed
WO-2005016918-A2 HETEROCYCLIC N-ARYL CARBOXAMIDES AS CYTOKINE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-02-24 WO claimed