SCHEMBL5690673

SCHEMBL5690673

Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(N3CCCC3)cc2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.65
ITGB1 P05556 3/20 0.47
ITGA5 P08648 3/20 0.47
L3MBTL1 Q9Y468 4/20 0.47
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
FKBP1A P62942 4/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 2/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.44
ITGAV P06756 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163529 0.94 ITGA4 (0.67) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL3860100 0.94 ITGA4 (0.67) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL6712483 0.91 ITGA4 (0.57) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL7071151 0.90 ITGA4 (0.58) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL5690767 0.90 ITGA4 (0.54) ITGA4ITGB1ITGA5L3MBTL1ITGAV
SCHEMBL7314087 0.89 ITGA4 (0.57) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL5690347 0.88 ITGA4 (0.75) ITGA4ITGB1ITGA5L3MBTL1GAA
SCHEMBL3848814 0.88 ITGA4 (0.53) ITGA4ITGB1ITGA5GAAHPGD
SCHEMBL3851600 0.87 ITGA4 (0.59) ITGA4ITGB1ITGA5GAAFKBP1A
SCHEMBL3857921 0.87 ITGA4 (0.54) ITGA4ITGB1ITGA5GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001974-B1 4-AMINO-PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2006-05-24 EP claimed
EP-1001974-B1 4-AMINO-PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2006-05-24 EP disclosed
US-6291453-B1 4-amino-phenylalanine type compounds which inhibit leukocyte adhesion mediated by VLA-4 ATHENA NEUROSCIENCES, INC. 2001-09-18 US disclosed