SCHEMBL5690772

SCHEMBL5690772

CC(=O)Nc1cccc(-c2ccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C3CC3)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 9/20 0.56
CYP3A4 P08684 3/20 0.56
PTGIR P43119 6/20 0.42
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NQO2 P16083 2/20 0.40
PIP5K1C O60331 1/20 0.39
PIK3CA P42336 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689071 0.86 CYP17A1 (0.52) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5689005 0.84 CYP17A1 (0.55) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5688994 0.84 CYP17A1 (0.55) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5690750 0.81 CYP17A1 (0.46) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5688825 0.81 CYP17A1 (0.45) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5690727 0.81 CYP17A1 (0.47) CYP17A1CYP3A4NPC1TSHRRAB9A
SCHEMBL5688534 0.78 CYP17A1 (0.67) CYP17A1CYP3A4PTGIRNPC1RAB9A
SCHEMBL5688963 0.78 CYP17A1 (0.45) CYP17A1CYP3A4PTGIRNPC1TSHR
SCHEMBL5688259 0.76 CYP17A1 (0.50) CYP17A1CYP3A4NPC1RAB9ASMN1; SMN2
SCHEMBL5688983 0.75 CYP3A4 (0.44) CYP17A1CYP3A4NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed