SCHEMBL5694965

SCHEMBL5694965

COC[C@H]1O[C@@H](n2cnc3c(NCCc4ccccc4)nc(CNS(=O)(=O)c4ccccc4)nc32)[C@@H](O)[C@@H]1O

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.58
PGK1 P00558 3/20 0.58
PGK2 P07205 3/20 0.58
NT5E P21589 5/20 0.58
ADORA3 P0DMS8 4/20 0.54
ADORA1 P30542 3/20 0.53
NFKB1 P19838 1/20 0.53
THPO P40225 1/20 0.53
TSHR P16473 1/20 0.53
ADORA2B P29275 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5694961 1.00 ADORA2A (0.58) ADORA2APGK1PGK2NT5EADORA3
SCHEMBL6328795 0.91 PGK1 (0.71) ADORA2APGK1PGK2NT5EADORA3
SCHEMBL6328801 0.91 PGK1 (0.71) ADORA2APGK1PGK2NT5EADORA3
SCHEMBL5695127 0.89 ADORA2A (0.72) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL5695133 0.89 ADORA2A (0.72) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL7771098 0.87 PGK1 (0.64) ADORA2APGK1PGK2NT5EADORA3
SCHEMBL5694952 0.87 PGK1 (0.64) ADORA2APGK1PGK2NT5EADORA3
SCHEMBL5695048 0.85 ADORA2A (0.74) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL5695041 0.85 ADORA2A (0.74) ADORA2ANT5EADORA3ADORA1ADORA2B
SCHEMBL5694948 0.84 ADORA2A (0.81) ADORA2APGK1PGK2NT5EADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1121372-B1 ADENINE DERIVATIVES PFIZER LTD (GB) 2006-06-28 EP disclosed
US-6326359-B1 PURINE DERIVATIVES PFIZER INC 2001-12-04 US disclosed