SCHEMBL5694952

SCHEMBL5694952

COC[C@H]1O[C@@H](n2cnc3c(NCCc4ccccc4)nc(CN)nc32)[C@H](O)[C@@H]1O

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 3/20 0.64
PGK2 P07205 3/20 0.64
ADORA2A P29274 8/20 0.63
NT5E P21589 2/20 0.61
ADORA3 P0DMS8 7/20 0.59
ADORA1 P30542 5/20 0.59
NFKB1 P19838 1/20 0.59
THPO P40225 1/20 0.59
TSHR P16473 1/20 0.59
ADORA2B P29275 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7771098 1.00 PGK1 (0.64) PGK1PGK2ADORA2ANT5EADORA3
SCHEMBL7049149 0.90 PGK1 (0.79) PGK1PGK2ADORA2AADORA3ADORA1
SCHEMBL5694942 0.88 ADORA2A (0.75) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL5695147 0.88 ADORA2A (0.75) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7777196 0.88 ADORA2A (0.75) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL5694965 0.87 ADORA2A (0.58) PGK1PGK2ADORA2ANT5EADORA3
SCHEMBL5694961 0.87 ADORA2A (0.58) PGK1PGK2ADORA2ANT5EADORA3
SCHEMBL5694960 0.87 PGK1 (0.64) PGK1PGK2ADORA2ANT5EADORA3
SCHEMBL5694954 0.87 PGK1 (0.64) PGK1PGK2ADORA2ANT5EADORA3
SCHEMBL5694948 0.86 ADORA2A (0.81) PGK1PGK2ADORA2ANT5EADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1121372-B1 ADENINE DERIVATIVES PFIZER LTD (GB) 2006-06-28 EP disclosed
US-6326359-B1 PURINE DERIVATIVES PFIZER INC 2001-12-04 US disclosed
EP-1121372-A1 ADENINE DERIVATIVES Pfizer Limited (GB) 2001-08-08 EP disclosed
WO-2000023457-A1 ADENINE DERIVATIVES PFIZER LIMITED (GB) 2000-04-27 WO disclosed