SCHEMBL5696407

SCHEMBL5696407

CCc1ccc(OCC(=O)Nc2ccccc2C(=O)O)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.76
TSHR P16473 2/20 0.67
MAPK10 P53779 2/20 0.67
ALDH1A1 P00352 2/20 0.67
HSD17B10 Q99714 1/20 0.67
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
CASP3 P42574 1/20 0.67
SENP8 Q96LD8 1/20 0.67
SENP7 Q9BQF6 1/20 0.67
SENP6 Q9GZR1 1/20 0.67
L3MBTL1 Q9Y468 2/20 0.63
LMNA P02545 1/20 0.63
KDM4E B2RXH2 3/20 0.63
POLB P06746 1/20 0.63
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
HIF1A Q16665 1/20 0.60
EPAS1 Q99814 1/20 0.60
MAPK1 P28482 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696414 0.90 HCAR2 (0.73) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL6032429 0.87 HCAR2 (0.81) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL18510324 0.86 NPC1 (0.80) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL8689332 0.86 HCAR2 (1.00) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL8943790 0.86 HCAR2 (0.79) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL5696427 0.85 HCAR2 (0.78) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL4914608 0.84 HCAR2 (0.76) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL4912964 0.84 NPC1 (0.80) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL4915695 0.84 HCAR2 (0.76) HCAR2TSHRMAPK10ALDH1A1HSD17B10
SCHEMBL4650500 0.83 HCAR2 (0.57) HCAR2TSHRMAPK10ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670749-A1 2-SUBSTITUTED BENZOIC ACID DERIVATIVES AS HM74A RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2006-06-21 EP disclosed
WO-2005016870-A1 2-SUBSTITUTED BENZOIC ACID DERIVATIVES AS HM74A RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-02-24 WO disclosed