SCHEMBL6032429

SCHEMBL6032429

O=C(COc1ccccc1)Nc1ccccc1C(=O)O

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.81
MAPK10 P53779 3/20 0.76
TSHR P16473 2/20 0.76
ALDH1A1 P00352 2/20 0.76
HSD17B10 Q99714 1/20 0.76
KMT2A Q03164 3/20 0.74
MEN1 O00255 2/20 0.74
CASP3 P42574 1/20 0.74
SENP8 Q96LD8 1/20 0.74
SENP7 Q9BQF6 1/20 0.74
SENP6 Q9GZR1 1/20 0.74
NPC1 O15118 5/20 0.68
RAB9A P51151 4/20 0.68
KDM4E B2RXH2 4/20 0.66
POLB P06746 2/20 0.66
L3MBTL1 Q9Y468 1/20 0.66
HIF1A Q16665 1/20 0.65
EPAS1 Q99814 1/20 0.65
TP53 P04637 1/20 0.59
RECQL P46063 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8943790 0.98 HCAR2 (0.79) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL5696427 0.91 HCAR2 (0.78) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL4912964 0.90 NPC1 (0.80) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL18510324 0.90 NPC1 (0.80) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL4914608 0.90 HCAR2 (0.76) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL4915695 0.90 HCAR2 (0.76) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL8689332 0.90 HCAR2 (1.00) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL14449495 0.89 HCAR2 (0.77) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL11597574 0.88 MAPK10 (0.72) HCAR2MAPK10TSHRALDH1A1HSD17B10
SCHEMBL5696407 0.87 HCAR2 (0.76) HCAR2MAPK10TSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7179411-A None JP disclosed
US-11691983-B2 Specifically substituted benzofuro- and benzothienoquinolines for organic light emitting diodes IDEMITSU KOSAN CO., LTD. (JP) 2023-07-04 US disclosed
US-11691983-B2 Specifically substituted benzofuro- and benzothienoquinolines for organic light emitting diodes IDEMITSU KOSAN CO., LTD. (JP) 2023-07-04 US disclosed
US-20190161497-A1 SPECIFICALLY SUBSTITUTED BENZOFURO- AND BENZOTHIENOQUINOLINES FOR ORGANIC LIGHT EMITTING DIODES IDEMITSU KOSAN CO., LTD. (JP) 2019-05-30 US disclosed
WO-2011057110-A1 GPR109A AGONISTS FOR THE TREATMENT OF CEREBRAL ISCHEMIA RUPRECHT-KARLS-UNIVERSITAT-HEIDELBERG (DE) 2011-05-12 WO disclosed
US-20110065676-A1 COMBINATION THERAPIES COMPRISING PAR1 ANTAGONISTS WITH NAR AGONISTS SCHERING CORPORATION (US) 2011-03-17 US disclosed
EP-1656139-A1 ARYL DICARBOXAMIDES Applied Research Systems ARS Holding N.V. (AN) 2006-05-17 EP disclosed
WO-2005011685-A1 ARYL DICARBOXAMIDES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (NL) 2005-02-10 WO disclosed
US-5925647-A TREATMENT OF INSULIN NON-INSULIN DEPENDENT DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5741926-A ANTIDIABETIC AGENT SHAMAN PHARMACEUTICALS, INC. (US) 1998-04-21 US disclosed
US-5681958-A TREATMENT OF DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1997-10-28 US disclosed
WO-1997030019-A1 ANILINE DERIVATIVES HAVING ANTIHYPERGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1997-08-21 WO disclosed
WO-1996010015-A1 CRYPTOLEPINE ANALOGS WITH HYPOGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1996-04-04 WO disclosed
JP-H07179411-A CRYSTAL OF BENZOIC ACID DERIVATIVE AND POLYVALENT METAL SALT OF THE BENZOIC ACID DERIVATIVE MITSUI TOATSU CHEM INC 1995-07-18 JP disclosed
EP-0376166-A1 Condensed quinoline system compound and process of preparation thereof MECT CORPORATION (JP) 1990-07-04 EP disclosed
EP-0364493-A1 RENIN INHIBITING PEPTIDES WITH NONPEPTIDE LINKAGES THE UPJOHN COMPANY (US) 1990-04-25 EP disclosed
WO-1989001488-A1 RENIN INHIBITING PEPTIDES WITH NONPEPTIDE LINKAGES THE UPJOHN COMPANY (US) 1989-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11691983-B2 Specifically substituted benzofuro- and benzothienoquinolines for organic light emitting diodes KCNQ2, KCNQ1, KCNQ4 HCAR2 2204/4885MAPK10 3518/4885TSHR 2470/4885
US-20190161497-A1 SPECIFICALLY SUBSTITUTED BENZOFURO- AND BENZOTHIENOQUINOLINES FOR ORGANIC LIGHT EMITTING DIODES KCNQ2, KCNQ1, KCNQ4 HCAR2 2204/4885MAPK10 3518/4885TSHR 2470/4885
US-20110065676-A1 COMBINATION THERAPIES COMPRISING PAR1 ANTAGONISTS WITH NAR AGONISTS F2R, F2RL1, F2RL3 HCAR2 97/4885MAPK10 2100/4885TSHR 1925/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.