SCHEMBL5697482

SCHEMBL5697482

Nc1ccnc(N)c1C(=O)NCc1ccc(Oc2cccc(F)c2)s1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LOX P28300 2/20 0.37
LOXL2 Q9Y4K0 2/20 0.37
PIN1 Q13526 2/20 0.37
KLKB1 P03952 5/20 0.37
GCK P35557 1/20 0.36
SLC8A1 P32418 2/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 1/20 0.35
HIF1A Q16665 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5697501 0.88 MAPK14 (0.40) GCK
SCHEMBL1680815 0.85 PDPK1 (0.41) ADORA2AADORA1
SCHEMBL1681150 0.83 KDM5A (0.41) LOXLOXL2KLKB1ADORA2AADORA1
SCHEMBL1681092 0.80 KLKB1 (0.41) LOXLOXL2PIN1KLKB1GCK
SCHEMBL1680495 0.80 KLKB1 (0.44) LOXLOXL2PIN1KLKB1SLC8A1
SCHEMBL1680873 0.78 POLB (0.42) LOXLOXL2ADORA2AALDH1A1
SCHEMBL14534354 0.78 PDPK1 (0.35) GCKNPSR1ALDH1A1
SCHEMBL1680964 0.76 SLC8A1 (0.45) KLKB1GCKSLC8A1
SCHEMBL12352596 0.76 SCN9A (0.41) PIN1GCKADORA2AADORA1NPSR1
SCHEMBL1680976 0.76 EGLN1 (0.47) LOXLOXL2KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1669348-A1 NOVEL ANTIFUNGAL AGENT COMPRISING HETEROCYCLIC COMPOUND Eisai Co., Ltd. (JP) 2006-06-14 EP disclosed