Fluoride

Fluoride

SCHEMBL5698381

Clc1ccc(SNc2ccccc2)cc1.F.F.F

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 1/20 0.40
TSHR P16473 1/20 0.40
CYP1A2 P05177 2/20 0.39
MAPT P10636 6/20 0.39
CNR1 P21554 4/20 0.39
PTGS2 P35354 1/20 0.38
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
IDO1 P14902 1/20 0.37
HPGD P15428 1/20 0.37
CHRNA7 P36544 1/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 2/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311562 0.82 HSD17B10 (0.50) TSHRCYP1A2MAPTPTGS2ALDH1A1
SCHEMBL18457231 0.78 CNR1 (0.42) CYP1A2CNR1ALDH1A1SMN1; SMN2LMNA
SCHEMBL24986294 0.77 HSD17B10 (0.35) TSHRCYP1A2MAPTPTGS2ALDH1A1
SCHEMBL11289053 0.77 HPGD (0.52) TSHRCYP1A2MAPTALDH1A1SMN1; SMN2
SCHEMBL26191084 0.77 MAOA (0.48) MAPTCNR1ALDH1A1SMN1; SMN2LMNA
SCHEMBL24124200 0.77 MAPT (0.52) TSHRCYP1A2MAPTPTGS2ALDH1A1
SCHEMBL7181962 0.77 MAOA (0.50) TSHRSMN1; SMN2LMNAIDO1RAB9A
SCHEMBL7181957 0.77 SMN1; SMN2 (0.38) TSHRCYP1A2MAPTPTGS2ALDH1A1
SCHEMBL6422226 0.76 NPC1 (0.49) CYP1A2MAPTALDH1A1LMNAIDO1
SCHEMBL3330967 0.74 MAOA (0.43) TSHRMAPTPTGS2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275631-B1 Fluorination with aminosulfur trifluorides AIR PROD & CHEM (US) 2006-07-19 EP disclosed
EP-1275631-A2 Fluorination with aminosulfur trifluorides AIR PRODUCTS AND CHEMICALS, INC. (US) 2003-01-15 EP disclosed
EP-0908448-B1 Thermally stable aminosulfur trifluorides AIR PROD & CHEM (US) 2001-11-14 EP disclosed
US-6242645-B1 BIOLOGICAL ACTIVITY ENHANCER, DEOXOFLUORINATION AGENT OF INTEREST IN MEDICINAL AND AGROCHEMICAL PRODUCTS AIR PRODUCTS AND CHEMICALS, INC. 2001-06-05 US disclosed
US-6222064-B1 PERFORMING FLUORINATION BY CONTACTING ALCOHOLS, ALDEHYDES, KETONES, EPOXIDES, AND MIXTURES USING A FLUORINATING REAGENT COMPRISING AMINOSULFUR TRIFLUORIDE COMPOUND AIR PRODUCTS AND CHEMICALS, INC. 2001-04-24 US disclosed
US-6207860-B1 FLUORINATING AGENTS, FAR LESS POTENTIAL OF VIOLENT DECOMPOSITION AND ATTENDANT HIGH GASEOUS BY-PRODUCT EVOLVEMENT, USEFUL FOR DEOXOFLUORINATION OF ALCOHOLS AND KETONES, AIR PRODUCTS AND CHEMICALS, INC. 2001-03-27 US disclosed
US-6080886-A STABLE, EFFICIENT FLUORINATION WITH LESS POTENTIAL OF VIOLENT DECOMPOSITION AND ATTENDANT HIGH GASEOUS BY-PRODUCT EVOLVEMENT; PRODUCING SYNTHETIC DRUGS AND AGROCHEMICAL PRODUCTS AIR PRODUCTS AND CHEMICALS, INC. (US) 2000-06-27 US disclosed
EP-0908448-A1 Thermally stable aminosulfur trifluorides AIR PRODUCTS AND CHEMICALS, INC. (US) 1999-04-14 EP disclosed
EP-0905109-A1 Fluorination with aminosulfur trifluorides AIR PRODUCTS AND CHEMICALS, INC. (US) 1999-03-31 EP disclosed