SCHEMBL5698592

SCHEMBL5698592

CS(=O)(=O)c1ccc(-c2cncn2-c2ccncc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.52
PTGS2 P35354 15/20 0.51
TDO2 P48775 1/20 0.51
MELK Q14680 1/20 0.48
PTGS1 P23219 4/20 0.44
FLT3 P36888 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6289849 0.87 PTGS2 (0.59) IDO1PTGS2TDO2PTGS1
SCHEMBL6294248 0.86 PTGS2 (0.63) IDO1PTGS2TDO2PTGS1
SCHEMBL6291198 0.86 PTGS2 (0.60) IDO1PTGS2PTGS1
SCHEMBL6180979 0.86 PTGS2 (0.63) IDO1PTGS2TDO2PTGS1
SCHEMBL6291219 0.85 PTGS2 (0.58) IDO1PTGS2TDO2PTGS1
SCHEMBL6293882 0.85 IDO1 (0.49) IDO1PTGS2TDO2PTGS1
SCHEMBL6291197 0.83 PTGS2 (0.62) IDO1PTGS2TDO2PTGS1
SCHEMBL6291082 0.83 PTGS2 (0.62) IDO1PTGS2TDO2PTGS1
SCHEMBL6291235 0.83 PTGS2 (0.59) IDO1PTGS2TDO2PTGS1
SCHEMBL6178888 0.82 IDO1 (0.47) IDO1PTGS2TDO2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682143-A2 COMBINATIONS COMPRISING AN HSP90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA Pharmacia Corporation (US) 2006-07-26 EP disclosed
WO-2005044194-A2 TREATMENT OR PREVENTION OF NEOPLASIA BY USE OF AN Hsp90 INHIBITOR PHARMACIA CORPORATION (US) 2005-05-19 WO disclosed
WO-2005041879-A2 COMBINATIONS COMPRISING AN Hsp90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed