SCHEMBL5698692

SCHEMBL5698692

Cc1cc(-c2ccc(S(N)(=O)=O)cc2)nn1-c1ccc(Cl)cc1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.70
PTGS1 P23219 4/20 0.66
CHRNA7 P36544 3/20 0.66
CYP2C9 P11712 1/20 0.58
PDPK1 O15530 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698697 0.85 PTGS2 (0.88) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL212983 0.85 PTGS2 (0.83) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8121503 0.85 PTGS2 (0.83) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8119233 0.83 PTGS2 (0.72) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8119412 0.83 PTGS2 (0.76) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8126281 0.82 PTGS2 (0.71) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8123558 0.82 PTGS2 (0.74) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8126311 0.82 PTGS2 (0.77) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8119016 0.81 PTGS2 (0.72) PTGS2PTGS1CHRNA7CYP2C9PDPK1
SCHEMBL8121094 0.81 PTGS2 (0.69) PTGS2PTGS1CHRNA7CYP2C9PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682143-A2 COMBINATIONS COMPRISING AN HSP90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA Pharmacia Corporation (US) 2006-07-26 EP disclosed
WO-2005044194-A2 TREATMENT OR PREVENTION OF NEOPLASIA BY USE OF AN Hsp90 INHIBITOR PHARMACIA CORPORATION (US) 2005-05-19 WO disclosed
WO-2005041879-A2 COMBINATIONS COMPRISING AN Hsp90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed