SCHEMBL5698707

SCHEMBL5698707

NS(=O)(=O)c1ccc(-c2oc(=O)[nH]c2-c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 8/20 0.54
CA1 P00915 6/20 0.54
CA9 Q16790 6/20 0.54
CA12 O43570 5/20 0.54
PTGS2 P35354 10/20 0.52
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
TNKS O95271 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3490095 0.84 KDM4E (0.50) CA2CA1CA9CA12
SCHEMBL7090696 0.78 CA2 (0.66) CA2CA1CA9CA12PTGS2
SCHEMBL7278194 0.75 NOTUM (0.45)
SCHEMBL308881 0.73 CA2 (1.00) CA2CA1CA9CA12PTGS2
SCHEMBL6482321 0.73 CA2 (1.00) CA2CA1CA9CA12PTGS2
Hydrochloric Acid SCHEMBL30685243 0.71 CA2 (0.95) CA2CA1CA9CA12PTGS2
SCHEMBL11753299 0.71 NOTUM (0.44) PTGS2
SCHEMBL6342030 0.69 PTGS2 (1.00) PTGS2
SCHEMBL6342623 0.69 PTGS2 (1.00) PTGS2
SCHEMBL7090564 0.69 PTGS2 (0.60) CA2CA1CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682143-A2 COMBINATIONS COMPRISING AN HSP90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA Pharmacia Corporation (US) 2006-07-26 EP disclosed
WO-2005044194-A2 TREATMENT OR PREVENTION OF NEOPLASIA BY USE OF AN Hsp90 INHIBITOR PHARMACIA CORPORATION (US) 2005-05-19 WO disclosed
WO-2005041879-A2 COMBINATIONS COMPRISING AN Hsp90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed