SCHEMBL570574

SCHEMBL570574

c1cn(CC2CCCCC2)cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 1.00
HRH4 Q9H3N8 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
CYP19A1 P11511 11/20 0.46
TBXAS1 P24557 4/20 0.43
GAA P10253 1/20 0.42
QPCT Q16769 1/20 0.42
OGG1 O15527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11047040 1.00 CYP2B6 (1.00) CYP2B6HRH4HRH3CYP19A1TBXAS1
SCHEMBL11046868 1.00 CYP2B6 (1.00) CYP2B6HRH4HRH3CYP19A1TBXAS1
SCHEMBL20076324 1.00 CYP2B6 (1.00) CYP2B6HRH4HRH3CYP19A1TBXAS1
SCHEMBL11046639 1.00 CYP2B6 (1.00) CYP2B6HRH4HRH3CYP19A1TBXAS1
Water SCHEMBL29258020 0.98 CYP2B6 (0.96) CYP2B6HRH4HRH3CYP19A1TBXAS1
Hydrochloric Acid SCHEMBL11047046 0.98 CYP2B6 (0.96) CYP2B6HRH4HRH3CYP19A1TBXAS1
Iodide SCHEMBL16164466 0.98 CYP2B6 (0.96) CYP2B6HRH4HRH3CYP19A1TBXAS1
SCHEMBL11047050 0.98 CYP2B6 (0.96) CYP2B6HRH4HRH3CYP19A1TBXAS1
SCHEMBL11051252 0.94 CYP2B6 (0.89) CYP2B6CYP19A1TBXAS1
Oxalic Acid SCHEMBL11048695 0.90 CYP2B6 (0.81) CYP2B6CYP19A1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US claimed
WO-2012019093-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-02-09 WO claimed
EP-0000951-B1 PHARMACEUTICAL FORMULATIONS COMPRISING 1-SUBSTITUTED IMIDAZOLES, 1-SUBSTITUTED IMIDAZOLES AND 1-SUBSTITUTED IMIDAZOLES FOR USE IN THE TREATMENT OR PROPHYLAXIS OF THROMBO-EMBOLIC DISORDERS THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-23 EP claimed
US-4284641-A ANTITHROMBOEMBOLIC AGENT BURROUGHS WELLCOME CO. (US) 1981-08-18 US claimed
EP-0000951-A1 Pharmaceutical Formulations comprising 1-substituted imidazoles, 1-substituted imidazoles and 1-substituted imidazoles for use in the treatment or prophylaxis of thrombo-embolic disorders THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP claimed
EP-3307739-A1 NRF2 REGULATORS GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-04-18 EP disclosed
US-9598342-B2 Production of acetic acid with enhanced catalyst stability CELANESE INTERNATIONAL CORPORATION (US) 2017-03-21 US disclosed
WO-2016202253-A1 NRF2 REGULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2016-12-22 WO disclosed
CN-102387992-B Molecular sieve and correlation technique and structure directing agent 加利福尼亚技术学院 2016-07-06 CN disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-4591594-A INSULIN LOWERING AGENTS HOFFMANN-LA ROCHE INC. (US) 1986-05-27 US disclosed
US-4581370-A Antiarrhythmic imidazoliums SCHERING A.G. (DE) 1986-04-08 US disclosed
US-4500540-A DIETETICS HOFFMANN-LA ROCHE INC. (US) 1985-02-19 US disclosed
EP-0131302-A2 Imidazolium salts, intermediates thereto and their use SCHERING AKTIENGESELLSCHAFT (DE) 1985-01-16 EP disclosed
EP-0000951-B1 PHARMACEUTICAL FORMULATIONS COMPRISING 1-SUBSTITUTED IMIDAZOLES, 1-SUBSTITUTED IMIDAZOLES AND 1-SUBSTITUTED IMIDAZOLES FOR USE IN THE TREATMENT OR PROPHYLAXIS OF THROMBO-EMBOLIC DISORDERS THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-23 EP disclosed
EP-0000950-B1 IMIDAZOLE DERIVATIVES AND SALTS THEREOF AND THEIR SYNTHESIS THE WELLCOME FOUNDATION LIMITED (GB) 1984-02-01 EP disclosed
US-4284641-A ANTITHROMBOEMBOLIC AGENT BURROUGHS WELLCOME CO. (US) 1981-08-18 US disclosed
EP-0000951-A1 Pharmaceutical Formulations comprising 1-substituted imidazoles, 1-substituted imidazoles and 1-substituted imidazoles for use in the treatment or prophylaxis of thrombo-embolic disorders THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION SLC6A3, NNT, SLC6A2 CYP2B6 902/4885HRH4 751/4885HRH3 998/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.