SCHEMBL5706141

SCHEMBL5706141

N=C(Cc1ccccc1)C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.54
CES2 O00748 1/20 0.54
AKR1B1 P15121 1/20 0.54
PLAU P00749 1/20 0.49
HIF1A Q16665 1/20 0.48
IDO1 P14902 3/20 0.47
NOS1 P29475 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
NOS3 P29474 1/20 0.47
NOS2 P35228 1/20 0.47
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45
F2 P00734 1/20 0.44
PLG P00747 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
C1S P09871 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621531 0.82 CES1 (0.58) CES1CES2AKR1B1PLAUMEN1
Phenylacetic Acid SCHEMBL27804643 0.80 AKR1B1 (0.77) CES1CES2AKR1B1PLAUHIF1A
Bicarbonate SCHEMBL6989215 0.80 CES1 (0.56) CES1CES2AKR1B1PLAUHIF1A
Phenylacetic Acid SCHEMBL28326941 0.78 AKR1B1 (0.74) CES1CES2AKR1B1PLAUHIF1A
SCHEMBL4461405 0.77 PRSS1 (0.61) PLAUF2PLGPRSS1PRSS2
SCHEMBL5188950 0.77 CES1 (0.73) CES1CES2AKR1B1HIF1AMEN1
SCHEMBL10584878 0.77 CES1 (0.58) CES1CES2AKR1B1HIF1AMEN1
SCHEMBL10584888 0.77 CES1 (0.58) CES1CES2AKR1B1HIF1AMEN1
Acetic Acid SCHEMBL3665413 0.77 CES1 (0.52) CES1CES2AKR1B1PLAUHIF1A
SCHEMBL25676 0.77 CES1 (0.64) CES1CES2AKR1B1HIF1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697309-B1 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF SE (DE) 2014-04-23 EP claimed
EP-1716120-A1 HERBICIDAL HETEROAROYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2006-11-02 EP claimed
EP-1697309-A2 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2006-09-06 EP claimed
WO-2005061443-A2 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-07-07 WO claimed
WO-2005061464-A1 HERBICIDAL HETEROAROYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-07-07 WO claimed
EP-2427451-B1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CO LTD (JP) 2019-03-20 EP disclosed
EP-1697309-B1 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF SE (DE) 2014-04-23 EP disclosed
EP-1716120-A1 HERBICIDAL HETEROAROYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2006-11-02 EP disclosed
EP-1697309-A2 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2006-09-06 EP disclosed
WO-2005061464-A1 HERBICIDAL HETEROAROYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-07-07 WO disclosed
WO-2005061443-A2 BENZOYL-SUBSTITUTED PHENYLALANINE AMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-07-07 WO disclosed