SCHEMBL5708205

SCHEMBL5708205

Cc1[c]c(SCc2cccc3cn(-c4ccc(C(F)(F)F)cc4)nc23)ccc1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.35
PARP2 Q9UGN5 7/20 0.35
PARP3 Q9Y6F1 7/20 0.35
ADORA3 P0DMS8 3/20 0.35
MPO P05164 1/20 0.35
NOTUM Q6P988 1/20 0.31
KDM1A O60341 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5708231 0.80 CRBN (0.36) MPOKDM1AKCNH2
SCHEMBL5708177 0.78 NR3C1 (0.35) MPO
SCHEMBL3968483 0.75 ADORA3 (0.43) PARP1PARP2PARP3ADORA3NOTUM
SCHEMBL3962929 0.73 PARP1 (0.45) PARP1PARP2PARP3ADORA3NOTUM
SCHEMBL3968503 0.73 NOTUM (0.43) PARP1PARP2PARP3ADORA3NOTUM
SCHEMBL3965152 0.72 PPARD (0.57)
SCHEMBL3961112 0.72 PPARD (0.41) PARP1
SCHEMBL3963602 0.72 ADORA3 (0.40) PARP1PARP2PARP3ADORA3NOTUM
SCHEMBL5708193 0.72 PARP1 (0.34) PARP1PARP2PARP3ADORA3NOTUM
SCHEMBL3966971 0.72 PPARA (0.48) PARP1PARP2PARP3ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706386-A1 BICYCLIC DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2006-10-04 EP claimed
WO-2005066136-A1 BICYCLIC DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-07-21 WO claimed