Oxyquinoline

Oxyquinoline

SCHEMBL5710199

OB(c1ccc(Cl)cc1F)c1ccc(Cl)cc1F.Oc1cccc2cccnc12

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.54
CHRM1 P11229 1/20 0.54
TSHR P16473 1/20 0.54
COMT P21964 1/20 0.54
ADRA1A P35348 1/20 0.54
METAP2 P50579 1/20 0.54
METAP1 P53582 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
KDM4E B2RXH2 5/20 0.48
ALOX12 P18054 2/20 0.48
SLC40A1 Q9NP59 4/20 0.46
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
CASP6 P55212 1/20 0.44
KDR P35968 2/20 0.44
LMNA P02545 4/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 3/20 0.42
MPI P34949 1/20 0.42
MAPT P10636 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxyquinoline SCHEMBL5163066 0.90 MMP2 (0.46) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL5165934 0.80 MMP2 (0.48) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL5167730 0.78 MMP2 (0.49) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL5164457 0.78 MMP2 (0.51) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL10787641 0.75 TSHR (0.88) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL29015237 0.75 TSHR (0.88) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL30367602 0.75 TSHR (0.95) MMP2CHRM1TSHRCOMTADRA1A
Oxyquinoline SCHEMBL29532359 0.75 TSHR (0.95) MMP2CHRM1TSHRCOMTADRA1A
SCHEMBL2404902 0.75 KMT2A (0.36) TSHRKMT2ALMNAALDH1A1NPC1
Oxyquinoline SCHEMBL543360 0.75 MMP2 (0.95) MMP2CHRM1TSHRCOMTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339725-B1 DNA METHYL TRANSFERASE INHIBITORS PENN STATE RES FOUND (US) 2006-11-22 EP disclosed