SCHEMBL571053

SCHEMBL571053

C=C(O[Si](C)(C)C(C)(C)C)C(=O)OCC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
TSHR P16473 1/20 0.40
DRD2 P14416 1/20 0.38
MGAM O43451 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 1/20 0.33
TRPA1 O75762 1/20 0.33
GLO1 Q04760 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
THRB P10828 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23461918 0.82 ALDH1A1 (0.33) ALDH1A1TSHRDRD2NPC1RAB9A
SCHEMBL28558851 0.82 ALDH1A1 (0.37) ALDH1A1TSHRDRD2MGAMGAA
SCHEMBL10644573 0.81 DRD2 (0.33) ALDH1A1TSHRDRD2MAPT
SCHEMBL9651307 0.81 DRD2 (0.35) ALDH1A1TSHRDRD2MAPT
SCHEMBL3534657 0.80 ALDH1A1 (0.45) ALDH1A1TSHRMGAMGAASI
SCHEMBL9703790 0.77 DRD2 (0.31) DRD2
SCHEMBL1879791 0.76 DRD2 (0.33) DRD2
SCHEMBL16316919 0.76 ALDH1A1 (0.50) ALDH1A1TSHRDRD2MGAMGAA
SCHEMBL14095603 0.76 GAA (0.58) ALDH1A1DRD2MGAMGAASI
SCHEMBL2219015 0.75 ALDH1A1 (0.38) ALDH1A1TSHRDRD2MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543263-B1 POLYOLEFIN-BASED EMULSIFIER AND APPLICATION THEREOF FOR PREPARING HIGH INTERNAL PHASE EMULSION AND POROUS POLYMERIC MATERIAL UNIV ZHEJIANG (CN) 2024-07-03 EP claimed
EP-3543263-A1 POLYOLEFIN-BASED EMULSIFIER AND APPLICATION THEREOF FOR PREPARING HIGH INTERNAL PHASE EMULSION AND POROUS POLYMERIC MATERIAL Zhejiang University (CN) 2019-09-25 EP claimed
EP-3543263-B1 POLYOLEFIN-BASED EMULSIFIER AND APPLICATION THEREOF FOR PREPARING HIGH INTERNAL PHASE EMULSION AND POROUS POLYMERIC MATERIAL UNIV ZHEJIANG (CN) 2024-07-03 EP disclosed
US-RE47741-E1 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2019-11-26 US disclosed
EP-3543263-A1 POLYOLEFIN-BASED EMULSIFIER AND APPLICATION THEREOF FOR PREPARING HIGH INTERNAL PHASE EMULSION AND POROUS POLYMERIC MATERIAL Zhejiang University (CN) 2019-09-25 EP disclosed
US-8658606-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-02-25 US disclosed
US-8653042-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-02-18 US disclosed
US-8524675-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-09-03 US disclosed
US-8524689-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-09-03 US disclosed
US-8492354-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-07-23 US disclosed
US-8481502-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-07-09 US disclosed
WO-2011044503-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
WO-2010132839-A2 AMINOGLYCOSIDE DOSING REGIMENS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132760-A1 ANTIBACTERIAL DERIVATIVES OF TOBRAMYCIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132759-A1 ANTIBACTERIAL DERIVATIVES OF DIBEKACIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132768-A1 ANTIBACTERIAL DERIVATIVES OF SISOMICIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132765-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132757-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010042851-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-04-15 WO disclosed
WO-2010042850-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-04-15 WO disclosed