SCHEMBL5717261

SCHEMBL5717261

PC(c1ccccc1)(c1ccccc1)C1CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
CHRM2 P08172 10/20 0.42
CHRM1 P11229 10/20 0.42
CHRM3 P20309 8/20 0.42
CHRM4 P08173 7/20 0.42
CHRM5 P08912 7/20 0.42
CYP2D6 P10635 4/20 0.42
KCNH2 Q12809 4/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
HRH1 P35367 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL11245316 0.98 KEAP1 (0.47) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL27838356 0.98 KEAP1 (0.50) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL9858885 0.93 KEAP1 (0.46) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL18788591 0.89 CYP2D6 (0.41) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL10907499 0.89 CYP2D6 (0.41) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL1403926 0.84 KEAP1 (0.50) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL3958141 0.82 KEAP1 (0.42) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL10448783 0.82 KEAP1 (0.42) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL5172183 0.82 KEAP1 (0.42) KEAP1NFE2L2CHRM2CHRM1CHRM3
SCHEMBL2464761 0.79 CYP2D6 (0.36) KEAP1NFE2L2CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678132-A1 PROCESS FOR THE PRODUCTION OF LACTAMS Davy Process Technology Limited (GB) 2006-07-12 EP claimed
WO-2005051907-A1 PROCESS FOR THE PRODUCTION OF LACTAMS DAVY PROCESS TECHNOLOGY LIMITED (GB) 2005-06-09 WO claimed