SCHEMBL5722142

SCHEMBL5722142

COc1ccc(CN2CCN(c3cc(Cl)nc(-n4ccnc4)n3)CC2C(=O)NCC2COc3ccccc3O2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 14/20 0.48
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.41
USP2 O75604 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5189774 0.90 ALDH1A1 (0.43) NOS2ALDH1A1KDM4EUSP2GLA
SCHEMBL7057672 0.84 NOS2 (0.42) NOS2ALDH1A1
SCHEMBL5192144 0.81 NOS2 (0.48) NOS2ALDH1A1KDM4EHPGDTSHR
SCHEMBL5191690 0.79 NOS2 (0.49) NOS2ALDH1A1KDM4EKMT2A
SCHEMBL6324458 0.78 NOS2 (0.70) NOS2
SCHEMBL5190808 0.78 NOS2 (0.65) NOS2
SCHEMBL5193371 0.77 NOS2 (0.66) NOS2
SCHEMBL5191424 0.77 ALDH1A1 (0.44) NOS2ALDH1A1USP2HPGDTSHR
SCHEMBL5211134 0.76 NOS2 (0.65) NOS2KDM4E
SCHEMBL5195036 0.76 NOS2 (0.54) NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LAB (US) 2006-11-15 EP disclosed