SCHEMBL5722162

SCHEMBL5722162

CC(=O)N1CCc2c([nH]c3ccc(Cl)cc23)C1c1ccc(O)cc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.66
KIF11 P52732 14/20 0.65
HTR2A P28223 2/20 0.56
HTR2C P28335 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.55
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13304608 0.95 SIRT1 (0.69) SIRT1KIF11ABCG2TP53MAPT
SCHEMBL3577188 0.89 KIF11 (0.80) KIF11
SCHEMBL11912895 0.89 KIF11 (0.59) SIRT1KIF11HTR2AHTR2CABCG2
SCHEMBL763586 0.87 KIF11 (0.58) SIRT1KIF11HTR2AHTR2CABCG2
SCHEMBL11912523 0.87 KIF11 (0.58) SIRT1KIF11HTR2AHTR2CABCG2
SCHEMBL764129 0.86 ABCG2 (0.63) SIRT1KIF11ABCG2TP53MAPT
SCHEMBL11912526 0.86 KIF11 (0.56) SIRT1KIF11HTR2AHTR2CABCG2
SCHEMBL3574031 0.86 KIF11 (0.66) SIRT1KIF11HTR2AHTR2C
SCHEMBL9962123 0.85 KIF11 (0.56) SIRT1KIF11HTR2AHTR2CABCG2
SCHEMBL8403284 0.85 KIF11 (0.56) SIRT1KIF11HTR2AHTR2CABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706404-A2 TETRAHYDROCARBOLINE COMPOUNDS AS ANTICANCER AGENTS Chiron Corporation (US) 2006-10-04 EP disclosed
WO-2005070930-A2 TETRAHYDROCARBOLINE COMPOUNDS AS ANTICANCER AGENTS CHIRON CORPORATION (US) 2005-08-04 WO disclosed