SCHEMBL5724601

SCHEMBL5724601

Cc1ccc(O)c(CC(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 1/20 0.52
HTT P42858 2/20 0.46
CSNK2A1 P68400 1/20 0.46
ALDH1A1 P00352 2/20 0.45
ALOX15 P16050 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TRPA1 O75762 1/20 0.45
ICMT O60725 3/20 0.44
CA2 P00918 1/20 0.44
TP53 P04637 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
ANO1 Q5XXA6 1/20 0.41
GAA P10253 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27745589 0.82 SRC (0.56) AMY1AHTTCSNK2A1ALOX15HSD17B10
SCHEMBL1478491 0.82 TAAR1 (0.52) HTTALDH1A1ICMTCA2TDP1
SCHEMBL30570712 0.82 TAAR1 (0.52) HTTALDH1A1ICMTCA2TDP1
SCHEMBL21363206 0.81 AMY1A (0.49) AMY1AHTTCSNK2A1ALDH1A1ALOX15
SCHEMBL28254697 0.81 ICMT (0.44) HTTALDH1A1ICMTCA2
SCHEMBL13068104 0.79 AMY1A (0.50) AMY1AHTTCSNK2A1ALDH1A1ALOX15
SCHEMBL10565369 0.79 ICMT (0.43) HTTALDH1A1ICMTCA2
SCHEMBL2702114 0.78 ICMT (0.45) HTTICMTCA2TP53TDP1
SCHEMBL5724612 0.78 CYP2D6 (0.57) ALDH1A1ALOX15HSD17B10TDP1ANO1
SCHEMBL7761752 0.78 SRC (0.56) ALDH1A1ALOX15ICMTGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8673897-B2 Benzodiazepinone compounds and methods of treatment using same THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2014-03-18 US disclosed
EP-1633715-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS Pfizer Limited (GB) 2006-03-15 EP disclosed
WO-2004108676-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS PFIZER LIMITED (GB) 2004-12-16 WO disclosed