SCHEMBL5725511

SCHEMBL5725511

CN(CCCC(c1ccc(F)cc1)c1ccc(F)cc1)C1CCCc2onc(O)c21

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.33
HTR2A P28223 1/20 0.30
HRH1 P35367 1/20 0.30
SCN5A Q14524 1/20 0.30
CCR5 P51681 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5725514 1.00 TBXA2R (0.33) TBXA2RHTR2AHRH1SCN5ACCR5
SCHEMBL8790520 1.00 TBXA2R (0.33) TBXA2RHTR2AHRH1SCN5ACCR5
SCHEMBL5724872 0.91 HTR2A (0.40) HTR2AHRH1CCR5
SCHEMBL5724916 0.85 CHRM2 (0.32)
SCHEMBL8790642 0.85 CHRM2 (0.32)
SCHEMBL5724742 0.81 KDM4E (0.34)
SCHEMBL5724739 0.81 KDM4E (0.34)
SCHEMBL5726294 0.78 SCN5A (0.38) SCN5A
SCHEMBL5726290 0.78 SCN5A (0.38) SCN5A
SCHEMBL5727812 0.75 HTR2A (0.37) HTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed
EP-0812318-A1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS H. LUNDBECK A/S (DK) 1997-12-17 EP disclosed
WO-1996026929-A1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS H. LUNDBECK A/S (DK) 1996-09-06 WO disclosed