SCHEMBL5726290

SCHEMBL5726290

Oc1noc2c1C(NCCCC(c1ccc(F)cc1)c1ccc(F)cc1)CCC2

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.38
VPS4B O75351 1/20 0.36
VCP P55072 1/20 0.36
ALDH1A1 P00352 2/20 0.34
CYP2C9 P11712 1/20 0.34
EPHX2 P34913 1/20 0.34
CACNA1B Q00975 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5726294 1.00 SCN5A (0.38) SCN5AVPS4BVCPALDH1A1CYP2C9
SCHEMBL5724914 0.83 SCN5A (0.35) SCN5AVPS4BVCPCYP2C9EPHX2
SCHEMBL5725809 0.80 DHODH (0.35) ALDH1A1MEN1KMT2A
SCHEMBL5725511 0.78 TBXA2R (0.33) SCN5A
SCHEMBL5725514 0.78 TBXA2R (0.33) SCN5A
SCHEMBL8790520 0.78 TBXA2R (0.33) SCN5A
SCHEMBL30674409 0.77 SCN5A (0.38) SCN5AVPS4BVCPALDH1A1CYP2C9
SCHEMBL5724732 0.77 DHODH (0.34) ALDH1A1MEN1KMT2A
SCHEMBL5726307 0.76 GRIN2B (0.44) ALDH1A1EPHX2
Bromide SCHEMBL5725876 0.76 LMNA (0.36) ALDH1A1CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed