SCHEMBL5725797

SCHEMBL5725797

CCOc1noc2c1[C@H](N(C)CCC=C(c1ccccc1C)c1ccccc1C)CCC2

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 8/20 0.34
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724743 0.87 SLC6A1 (0.36) SLC6A1
SCHEMBL5725795 0.80 SLC6A1 (0.34) SLC6A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL5725232 0.79 KDM4E (0.33) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5725226 0.79 KDM4E (0.33) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5725697 0.77 HRH1 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5727812 0.76 HTR2A (0.37) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5727815 0.76 HTR2A (0.37) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7979790 0.73 CHRM3 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7979788 0.73 CHRM3 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5725094 0.72 SLC6A1 (0.36) SLC6A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed